| ID |
Refrence |
Source Clone name |
Sequence |
Motif |
Target-tumor |
Target-cell |
Receptors-biomarker |
Phage/Library |
In vitro/Ex-vivo |
In vivo |
Homing/targeting |
Payloads |
Patent |
| 1009 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | E3 | YSINDWH | YSXNXW and PXNXXN | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | US2010/0233161A1 |
| 1010 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | B1 | YSFNSWM | YSXNXW | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | US2010/0233161A1 |
| 1011 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | D2 | PNPNNST | PXNXXN | Esophagus and gastroesophageal cancer | Tumor vessel | EGFR, EGFRvIII | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | US2010/0233161A1 |
| 1012 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | NA | YPTPYDI | NA | Esophagus and gastroesophageal cancer | Tumor vessel | Alpha-5 beta -5 integrins | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | US2010/0233161A1 |
| 1013 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | F1 | LPAMPNS | NA | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | NA |
| 1014 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | NA | CNRRTKAGC | NA | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | NA |
| 1015 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | NA | SRHDLNS | NA | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | NA |
| 1016 | Zhi M et al. Chin Med J (Engl). 2011 Feb;124(4):581-5. | NA | STVATSQ | NA | Esophagus and gastroesophageal cancer | Tumor vessel | NA | M13 phage/C7C peptide library | NA | 2-month-old Balb/c mice with human esophageal tumor xenograft, fresh human esophageal cancer tissue in immunosuppressed Balb/c mice | Homing | NA | NA |
| 1183 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CGKRK | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2006/0002854A1 |
| 1184 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CDTRL | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2006/0002854A1 |
| 1185 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CGTKRKC | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | NA |
| 1186 | Hoffman JA et al. Cancer Cell. 2003 Nov;4(5):383-91. | NA | CDTAVVEGL | NA | Epidermal squamous cell cancers | Tumor vessel | MECA32 (Second endothelial marker, the cell-surface antigen) | T7 phage /9-mer cyclic (CX7C) peptide library | NA | K14-HPV16 mice, FVB/b mice , C57B16 cells bearing mice,RIP1-Tag2 mice | Homing | NA | US 2011/0003848 A1 |
| 1190 | Rafii S et al. Cancer Cell. 2003 Nov;4(5):331-3. | NA | CRSRKG | NA | Pancreatic tumor | Tumor vessel | NA | T7 phage /9-mer cyclic (CX7C) peptide library | NA | RIP-Tag2 pancreatic tumors in murine model | Homing | NA | US 7,598,341 B2 |
| 1191 | Rafii S et al. Cancer Cell. 2003 Nov;4(5):331-3. | NA | CEYQLDVE | NA | Pancreatic tumor | Tumor vessel | NA | T7 phage /9-mer cyclic (CX7C) peptide library | NA | RIP-Tag2 pancreatic tumors in murine model | Homing | NA | US 7,598,341 B2 |
| 1322 | Karmali PP et al. Nanomedicine. 2009 Mar;5(1):73-82. | NA | CREKA | NA | Breast cancer | Tumor vessel | Clotted plasma proteins | NA | NA | Mice bearing MDA-MB-435 human cancer xenografts | Homing | Iron oxide nanoparticle,Abraxane | US20050048063 A1 |
| 1325 | Samanta S et al. Biomaterials. 2010 Mar;31(7):1787-97. | NA | CRGDGWC | RGD | Melanoma | Tumor vessel | Integrins Alpha- 5 beta -1 | NA | NA | Mice bearing the aggressive B16F10 tumor | Homing | NA | NA |
| 1326 | Samanta S et al. Biomaterials. 2010 Mar;31(7):1787-97. | RGDGWK-lipopeptide | RGDGWK | RGD | Melanoma | Tumor vessel | Integrins Alpha -5 beta- 1 | NA | NA | Mice bearing the aggressive B16F10 tumor | Homing | Anticancer-p-53 gene | NA |
| 1350 | Park JH et al. Small. 2009 Mar;5(6):694-700. | NA | CREKA | NA | Breast cancer ,Fibrosarcoma | Tumor vessel and stroma of tumors | NA | NA | NA | Mice bearing human (MDA-MB-435 human carcinoma and HT1080 human fibrosarcoma) xenograft | Homing | Superparamagnetic nanospheres, superparamagnetic IO nanoworms (NWs) | US20050048063A1 |
| 1373 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | PC5-52 | SVSVGMKPSPRP | PSP | Lung and Prostate cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice human cancers including human lung (H460), colon (HCT116), breast (BT483), prostate (PC3), liver (Mahlavu), and pancreatic (PaCa) cancer xenografts | Homing | Doxorubicin | US/ 20100119444A1,US 2010/0260673A1 |
| 1374 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | PC5-54 | WPLHTSVYPPSP | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing | NA | US 2008/0193510A1 |
| 1375 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-5 | NTLPPFSPPSPP | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1376 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-10 | SFPDSNIAPSSP | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1377 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-8 | QHAPSNSKSVLT | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1378 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-7 | WPTYLNPSSLKA | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1379 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-57 | GPSGNLHIRPAS | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1380 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-53 | SPLLSTRAVQLS | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1381 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-58 | SPMFTMIQGDAQ | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1382 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-60 | VNSHQALWSPAQ | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1383 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-4 | STLPPPLRFANV | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | US 2008/0193510A1 |
| 1384 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-2 | SFNQPYLYKTAF | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1385 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-3 | YHTRIALPDNLP | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1386 | Lee TY et al. Cancer Res. 2007 Nov 15;67(22):10958-65. | Clone PC5-11 | AQSTAFQKPLLM | NA | Lung cancer | Tumor vessel | Integrins, Alpha-5 beta-3 and Alpha-5 beta-5 | M13 phage/random peptide library | CL1-5 (lung cancer), H460 (lung cancer) ,PC-3 (prostate cancer),VEGF-stimulated HUVECs and human lung cancer vessels | SCID mice with lung cancer xenograft | Homing (Phage display clone) | NA | NA |
| 1396 | Maruta F et al. J Drug Target. 2007 May;15(4):311-9. | NA | VPNTNSLPAAVN | TNSLP | Human colorectal tumor | Tumor vessel | NA | M13 phage/12-mer linear peptide library | Human colorectal cancer biopsies | NA | Targeting | NA | NA |
| 1397 | Maruta F et al. J Drug Target. 2007 May;15(4):311-9. | NA | LIAKTALPQTNK | AxPxTN | Human colorectal tumor | Tumor vessel | NA | M13 phage/12-mer linear peptide library | Human colorectal cancer biopsies | NA | Targeting | NA | NA |
| 1399 | Maruta F et al. J Drug Target. 2007 May;15(4):311-9. | NA | LIAKTALPQTN | AxPxTN | Human colorectal tumor | Tumor vessel | NA | M13 phage/12-mer linear peptide library | Human colorectal cancer biopsies | NA | Targeting | NA | NA |
| 1468 | Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36. | NA | CVSNPRWKC | NA | Pancreatic islet tumors | Tumor vessel | EphA4, a receptor for epinephrine-A | Phage/ CX7C peptide library | EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cells | Male C57BL/6/RIP-Tag2 transgenic mice | Homing | NA | NA |
| 1469 | Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36. | NA | CHVLWSTRC | NA | Pancreatic islet tumors | Tumor vessel | EphA4, a receptor for epinephrine-A | Phage/ CX7C peptide library | EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cells | Male C57BL/6/RIP-Tag2 transgenic mice | Targeting | NA | NA |
| 1470 | Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36. | NA | SWLAYPGAVSYR | NA | Pancreatic islet tumors | Tumor vessel | Epinephrine-A | Phage/ CX7C peptide library | EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cells | Male C57BL/6/RIP-Tag2 transgenic mice | Targeting | NA | NA |
| 1471 | Yao VJ et al. Am J Pathol. 2005 Feb;166(2):625-36. | NA | YSAYPDSVPMMS | NA | Pancreatic islet tumors | Tumor vessel | Epinephrine-A | Phage/ CX7C peptide library | EphA2-Fc protein and to the EphA2 receptor expressed on human umbilical vein endothelial cells , MDA-MB-435 cultured human breast carcinoma cells | Male C57BL/6/RIP-Tag2 transgenic mice | Targeting | NA | NA |
| 1734 | NA | Clone 35 | VGVGEWSV | NA | Premalignant pancreas | Tumor vessel | NA | T7phage/(CX7C) peptide library | NA | RIP-Tag2 mice | Homing | Doxorubicin | US 2005/0245445A1 |
| 1735 | NA | Clone 1 | SRPRR | NA | Pre-malignant dysplastic skin | Tumor vessel | NA | T7phage/(CX7C) peptide library | NA | K14HPV16 mice bearing protuberant ear or trunk tumors at 9 to 12 months of age | Homing | Apoptotic peptide (KLAKLAK) | US 2011/0002848A1 |
| 1736 | NA | Clone 2 | CXSRPRRZC | NA | Pre-malignant dysplastic skin | Tumor vessel | NA | T7phage/(CX7C) peptide library | NA | K14HPV16 mice bearing protuberant ear or trunk tumors at 9 to 12 months of age | Homing | NA | US 2011/0002848A1 |
| 1737 | NA | NA | CSRPRRSVC | NA | Pre-malignant dysplastic skin | Tumor vessel | NA | NA | NA | K14HPV16 mice bearing protuberant ear or trunk tumors at 9 to 12 months of age | Homing | NA | US 2011/0002848A1 |
| 1738 | NA | NA | CSRPRRSWC | NA | Pre-malignant dysplastic skin | Tumor vessel | NA | NA | NA | K14HPV16 mice bearing protuberant ear or trunk tumors at 9 to 12 months of age | Homing | NA | US 2011/0002848A1 |
| 1753 | Lu ZX et al. Int J Nanomedicine 2011;6:1661-73. | APRPG peptide | APRPG | NA | Breast cancer | Tumor vessel | VEGF | NA | Human breast cancer cell line MCF-7 | BALB/C nude mice (5 weeks of age) | Homing | NA | US 6,753,310 B1 |
| 1756 | Numata K et al .Bioconjug Chem 2011 Aug 17;22(8):1605-10. | F3 | KDEPQRRSARLSAKPAPPKPEPKPKKAPAKK | NA | Breast tumor | Tumor vessel | Nucleolin | NA | MDA-MB-435 melanoma cell line, MDA-MB-231 | Mice bearing MDA-MB-231 | Homing | pDNA complexes of silk proteins containing poly(L-lysine) | US 7,544,767 B2 |
| 1757 | Numata K et al .Bioconjug Chem 2011 Aug 17;22(8):1605-10. | NA | CGKRK | NA | Breast tumor | Tumor vessel | Heparansulphate | NA | MDA-MB-435 melanoma cell line, MDA-MB-231 | Mice bearing MDA-MB-231 | Homing | pDNA complexes of silk proteins containing poly(L-lysine) | US 7,723,474 B2 |
| 1758 | Bhojani MS et al .PloS One. 2011;6(7):e22418. | Modified F3 | KDEPQRRSARLSAKPAPPKPEPKPKKAPAKKC | NA | Breast tumor | Tumor vessel | Nucleolin | NA | MDA-MB-435 melanoma cell line | Nude Mice bearing MDA-MB-435 | Homing | Radio idionated maleimide conjugating group | US 2005/0196343 A1 |